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Golden Packs

Golden Packs are pre-validated target bundles that include everything you need to start scoring: a prepared receptor grid, validated scoring profile, reference actives and decoys, and published benchmark results. They're the fastest way to get production-ready scoring on well-studied targets.

What's in a Golden Pack?

Each Golden Pack contains:

Component Description
Compiled Grid Pre-computed scoring grid ready for IsoDock/IsoScore
Scoring Profile Optimized weights validated against DEKOIS2
Reference Actives Known active compounds (SDF with 3D poses)
Reference Decoys Matched decoys from DEKOIS2
Benchmark Report AUC, enrichment factors, ROC curve, score distributions
Manifest Metadata including target class, tier, validation stats

Available Golden Packs

ACE Platinum Pack

Property Value
Target Angiotensin-converting enzyme
PDB 1O86
Class Metalloprotease
AUC 0.95
Tier Platinum
Actives 40
Decoys 1,200

ACE is a zinc metalloprotease critical in blood pressure regulation. The Platinum profile leverages metal coordination scoring and electrostatic complementarity.

Key profile features: Strong E_coul weight (0.22), metal coordination emphasis (0.18), moderate burial contribution.

MDM2 Gold Pack

Property Value
Target Mouse double minute 2 homolog
PDB 4HG7
Class Protein-protein interaction (PPI)
AUC 0.85
Tier Gold
Actives 78
Decoys 2,340

MDM2 is a key PPI target in oncology (p53-MDM2 interaction). The pocket is shallow and hydrophobic, requiring emphasis on shape complementarity and aromatic stacking.

Key profile features: High aromaticBurial weight, depth scoring, moderate dispersion.

CDK2 Silver Pack

Property Value
Target Cyclin-dependent kinase 2
PDB 1AQ1
Class Kinase
AUC 0.72
Tier Silver
Actives 219
Decoys 6,570

CDK2 is a well-studied kinase target. The Silver tier indicates moderate but useful discrimination, suitable for initial screening with additional validation recommended.

HSP90 Silver Pack

Property Value
Target Heat shock protein 90
PDB 2WI7
Class Chaperone
AUC 0.68
Tier Silver
Actives 88
Decoys 2,640

HSP90 is a molecular chaperone with a deep ATP-binding pocket. The Silver profile captures the key hydrogen bonding patterns in the pocket.

Using Golden Packs

Loading a Pack

  1. Go to Golden Packs in the sidebar
  2. Browse available packs by target or tier
  3. Click Load Pack to add it to your project
  4. The target, profile, and reference compounds are imported automatically

Scoring with a Golden Pack

Once loaded, the pack's target and profile are ready to use:

  1. Go to Workbench > IsoScore (or IsoDock)
  2. Select the Golden Pack target
  3. Upload your own ligands
  4. The optimized profile is automatically selected
  5. Click Run

Validating the Pack

To verify the pack works on your system:

  1. After loading, click Run Benchmark
  2. This scores the included reference actives and decoys
  3. Compare your AUC to the published value
  4. Results should match within +/- 0.02 AUC

Tip: Running the benchmark on your system is a good way to verify WebGPU performance and confirm everything is configured correctly.

Requesting New Packs

We're continuously expanding the Golden Packs library. Currently planned:

  • EGFR Kinase — in optimization pipeline
  • P38a Kinase — in optimization pipeline
  • HIVRT — Platinum profile available, pack assembly in progress

If you need a pack for a specific target, contact us at support@latticezero.com.

Building Your Own "Golden Pack"

While official Golden Packs are curated and validated, you can create your own validated bundles:

  1. Prepare your target using Target Prep
  2. Optimize a profile using the Optimizer with your known actives/decoys
  3. Validate by running the benchmark and checking AUC
  4. Save the target, profile, and reference compounds as a project

This is especially useful for proprietary targets where no official pack exists.

Next Steps